產(chǎn)品屬性:
產(chǎn)品名稱 | S26131 |
規(guī)格 | 1mg、5mg、10mg、25mg、50mg、100mg、200mg |
貨號(hào) | EY-01Y15057 |
Cas No.: 296280-56-3
別名: N/A
化學(xué)名: N/A
分子式: C31H34N2O4
分子量: 498.61
溶解度: DMSO: 5 mg/mL (10.03 mM)
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
S26131 (compound 5) is a potent and selective MT1 melatoninergic ligand, and the Ki values are 0.5 and 112 nM for MT1 and MT2, respectively. S26131 behaves as an MT1 and MT2 antagonist[1].S26131 behaves as an antagonist on MT1 and MT2 receptors with KB values of 5.32 and 143 nM, respectively[1].[1]. Descamps-Fran?ois C, et al. Design and synthesis of naphthalenic dimers as selective MT1 melatoninergic ligands. J Med Chem. 2003 Mar 27;46(7):1127-9.
特別提醒公司產(chǎn)品僅供科研使用