產(chǎn)品屬性：
產(chǎn)品名稱 | Salvinorin A Propionate |
規(guī)格 | 1mg、5mg、10mg |
貨號(hào) | EY-01Y14992 |
Cas No.: 689295-71-4
別名: N/A
化學(xué)名: N/A
分子式: C24H30O8
分子量: 446.5
溶解度: Acetonitrile: 1 mg/ml,DMF: 2 mg/ml,DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml,DMSO: 1 mg/ml
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述：
Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM. It inhibits adenylate cyclase (EC50 = 4.7 nM) in HEK293 cells transfected with human KOR. It is selective for KORs over μ, δ, and ORL-1 opioid receptors and has no effect at serotonin, dopamine, muscarinic, or adrenergic receptors. In mice, salvinorin A propionate (13 μg, i.c.v.) reduces nociceptive responses in a radiant heat tail-flick assay, though not as potently as salvinorin A .
特別提醒公司產(chǎn)品僅供科研使用
