產(chǎn)品屬性:
產(chǎn)品名稱(chēng) | Pemafibrate racemate |
規(guī)格 | 1mg、5mg、10mg、50mg、100mg |
貨號(hào) | EY-01Y14194 |
Cas No.: 848258-31-1
別名: N/A
化學(xué)名: N/A
分子式: C28H30N2O6
分子量: 490.55
溶解度: Soluble in DMSO
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
Pemafibrate racemate is the racemate of pemafibrate, and activates PPARα activity, with EC50s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively.
h-PPARα|1 nM (EC50)|h-PPARδ|1.7 μM (EC50)
Pemafibrate racemate activates PPARα activity, with EC50s of 1 nM, >10 μM and 1.7 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively[1].[1]. Yamazaki Y, et al. Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor alpha agonists. Bioorg Med Chem Lett. 2007 Aug 15;17(16):4689-93. Epub2007 May 24.
特別提醒公司產(chǎn)品僅供科研使用